Molecule Details
InChIKeyTWDZVSFDJAHALH-UHFFFAOYSA-N
Compound Name4-Benzoyl-1-(2-methyl-1-(2-oxopropyl)-1H-indol-4-yl)-5-phenyl-N-(5-sulfamoyl-1,3,4-thiadiazol-2-yl)-1H-pyrazole-3-carboxamide
Canonical SMILESCC(=O)Cn1c(C)cc2c(-n3nc(C(=O)Nc4nnc(S(N)(=O)=O)s4)c(C(=O)c4ccccc4)c3-c3ccccc3)cccc21
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.79
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P18505 GABRB1 Homo sapiens Human PF02931 PF02932 7.0 pIC50 TTD_MultiTarget
P00915 CA1 Homo sapiens Human PF00194 6.7 IC50 ChEMBL;BindingDB
P00918 CA2 Homo sapiens Human PF00194 6.7 IC50 ChEMBL;BindingDB