Molecule Details
InChIKeyTWBRLXCGQXCXSU-HCHGDIHTSA-N
Compound NameAdp[-Trp-Arg-Nva-Arg-Tyr-NH2]2
Canonical SMILESCCC[C@H](NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@@H](N)CC[C@H](N)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCC)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccc(O)cc1)C(N)=O)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccc(O)cc1)C(N)=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.22
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P50391 NPY4R Homo sapiens Human PF00001 8.4 Ki ChEMBL;BindingDB
P25929 NPY1R Homo sapiens Human PF00001 6.8 Ki ChEMBL;BindingDB
P49146 NPY2R Homo sapiens Human PF00001 6.4 Ki ChEMBL;BindingDB