Molecule Details
InChIKeyTUIRYRPRPHCOOR-UHFFFAOYSA-N
Compound Name1-[4-[2-(3-cyclopropyl-3-hydroxyazetidin-1-yl)ethoxy]-3-ethylphenyl]-4-(4-cyclopropylphenoxy)-2H-pyrrol-5-one
Canonical SMILESCCc1cc(N2CC=C(Oc3ccc(C4CC4)cc3)C2=O)ccc1OCCN1CC(O)(C2CC2)C1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.27
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q99705 MCHR1 Homo sapiens Human PF00001 9.4 Ki ChEMBL;BindingDB
P08684 CYP3A4 Homo sapiens Human PF00067 6.2 IC50 ChEMBL
P10635 CYP2D6 Homo sapiens Human PF00067 6.2 IC50 ChEMBL