Molecule Details
InChIKeySZBUKBINUVLFEL-UHFFFAOYSA-N
Compound Name4-amino-5-cyano-6-ethoxy-N-(pyridin-3-ylmethyl)pyridine-2-carboxamide
Canonical SMILESCCOc1nc(C(=O)NCc2cccnc2)cc(N)c1C#N
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.16
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P45983 MAPK8 Homo sapiens Human PF00069 7.6 IC50 ChEMBL;BindingDB
P45984 MAPK9 Homo sapiens Human PF00069 7.4 IC50 ChEMBL;BindingDB
P28482 MAPK1 Homo sapiens Human PF00069 6.5 Ki ChEMBL