Molecule Details
InChIKeySYNHRWSDSNIWGA-UHFFFAOYSA-N
Compound Name4-({2-[6-(1H-pyrazol-4-yl)-1H-indazol-3-yl]-1H-indol-5-yl}methyl)morpholine
Canonical SMILESc1cc2[nH]c(-c3n[nH]c4cc(-c5cn[nH]c5)ccc34)cc2cc1CN1CCOCC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.73
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O14757 CHEK1 Homo sapiens Human PF00069 8.0 IC50 ChEMBL;BindingDB
P50613 CDK7 Homo sapiens Human PF00069 7.6 IC50 ChEMBL
P51946 CCNH Homo sapiens Human PF16899 PF00134 7.6 IC50 BindingDB