Molecule Details
InChIKeySYCWRTUPLPDKDX-UHFFFAOYSA-N
Compound Name3-[6-(2-pyridin-2-yl-5,6-dihydro-4H-pyrrolo[2,1-e]pyrazol-3-yl)benzimidazol-1-yl]propan-1-ol
Canonical SMILESOCCCn1cnc2ccc(-c3c(-c4ccccn4)nn4c3CCC4)cc21
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.57
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P36897 TGFBR1 Homo sapiens Human PF01064 PF00069 PF08515 7.1 IC50 ChEMBL;BindingDB
P37173 TGFBR2 Homo sapiens Human PF08917 PF07714 6.5 IC50 ChEMBL;BindingDB
Q9NYL2 MAP3K20 Homo sapiens Human PF07714 PF07647 6.2 IC50 ChEMBL;BindingDB