Molecule Details
InChIKeySXWAEKQQXUUNDG-UHFFFAOYSA-N
Compound Name4-[4-[[2-[4-(4-Fluorophenyl)piperazin-1-yl]-6-methylpyrimidin-4-yl]oxymethyl]triazol-1-yl]benzenesulfonamide
Canonical SMILESCc1cc(OCc2cn(-c3ccc(S(N)(=O)=O)cc3)nn2)nc(N2CCN(c3ccc(F)cc3)CC2)n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.58
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P00918 CA2 Homo sapiens Human PF00194 9.1 Ki ChEMBL;BindingDB
O43570 CA12 Homo sapiens Human PF00194 7.3 Ki ChEMBL;BindingDB
Q16790 CA9 Homo sapiens Human PF00194 6.3 Ki ChEMBL;BindingDB