Molecule Details
InChIKeySXUNZFYJEHXSOJ-UHFFFAOYSA-N
Compound NameN-(2-aminoethyl)-4-(2-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl)benzenesulfonamide
Canonical SMILESCc1cc2c(-c3ccc(S(=O)(=O)NCCN)cc3)ccnc2[nH]1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.03
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O14920 IKBKB Homo sapiens Human PF18397 PF12179 PF00069 7.7 IC50 ChEMBL;BindingDB
O15111 CHUK Homo sapiens Human PF18397 PF12179 PF00069 6.9 IC50 ChEMBL;BindingDB
Q13464 ROCK1 Homo sapiens Human PF25346 PF00069 PF08912 6.5 IC50 ChEMBL;BindingDB