Molecule Details
InChIKeySXTDDUKKQSLXMI-UHFFFAOYSA-N
Compound Name6-(1-acetylazetidin-3-yl)sulfonyl-3-(2-amino-1H-benzimidazol-4-yl)-2-(2H-tetrazol-5-yl)benzenesulfonamide
Canonical SMILESCC(=O)N1CC(S(=O)(=O)c2ccc(-c3cccc4nc(N)[nH]c34)c(-c3nn[nH]n3)c2S(N)(=O)=O)C1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL9.24
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
C7C422 blaNDM-1 Klebsiella pneumoniae Pathogen PF00753 9.8 IC50 ChEMBL;BindingDB
Q9XAY4 blaVIM Pseudomonas aeruginosa Pathogen PF00753 9.4 IC50 BindingDB
P52699 Serratia marcescens Pathogen PF00753 8.6 IC50 BindingDB