Target not found.
Molecule Details
InChIKeySXJDVALQPLDIFB-KRWDZBQOSA-N
Compound Name(6S)-N-[(4-carbamimidoylphenyl)methyl]-1-chloro-3-(cyclobutylamino)-4-oxospiro[6,7-dihydropyrrolo[1,2-a]pyrazine-8,1'-cyclopentane]-6-carboxamide
Canonical SMILESN=C(N)c1ccc(CNC(=O)[C@@H]2CC3(CCCC3)c3c(Cl)nc(NC4CCC4)c(=O)n32)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.04
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P00734 F2 Homo sapiens Human PF00594 PF00051 PF09396 PF00089 7.1 Ki ChEMBL;BindingDB
P08709 F7 Homo sapiens Human PF00008 PF14670 PF00594 PF00089 7.0 Ki ChEMBL
P13726 F3 Homo sapiens Human PF09294 PF01108 7.0 Ki ChEMBL