Molecule Details
InChIKeySXCZVZBSIYFIES-UHFFFAOYSA-N
Compound Name5-{6-[4-(2-Bromo-5-fluorophenoxy)piperidin-1-yl]pyridazin-3-yl}nicotinic acid
Canonical SMILESO=C(O)c1cncc(-c2ccc(N3CCC(Oc4cc(F)ccc4Br)CC3)nn2)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Unknown
Avg pChEMBL8.28
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q86SK9 SCD5 Homo sapiens Human PF00487 8.4 IC50 ChEMBL;BindingDB
O00767 SCD Homo sapiens Human 8.2 IC50 ChEMBL;BindingDB