Molecule Details
InChIKeySWSOLWZGKLCZDP-UHFFFAOYSA-N
Compound Name4-{3-[2,2-Bis-(4-chloro-phenyl)-benzo[1,3]dioxole-5-carbonyl]-2-methyl-indol-1-yl}-butyric acid
Canonical SMILESCc1c(C(=O)c2ccc3c(c2)OC(c2ccc(Cl)cc2)(c2ccc(Cl)cc2)O3)c2ccccc2n1CCCC(=O)O
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL8.0
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P18405 SRD5A1 Homo sapiens Human PF02544 8.0 IC50 ChEMBL;BindingDB
P18505 GABRB1 Homo sapiens Human PF02931 PF02932 8.0 pIC50 TTD_MultiTarget
P31639 SLC5A2 Homo sapiens Human PF00474 8.0 pIC50 TTD_MultiTarget