Molecule Details
InChIKeySWQVIBOZAHRMDS-JXAWBTAJSA-N
Compound Name(Z)-3-(4-Oxo-2-{[2-oxo-5-(piperidin-1-ylsulfonyl)indolin-3-ylidene]methyl}-4,5,6,7-tetrahydro-1H-indol-3-yl)propanoic Acid
Canonical SMILESO=C(O)CCc1c(/C=C2\C(=O)Nc3ccc(S(=O)(=O)N4CCCCC4)cc32)[nH]c2c1C(=O)CCC2
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.33
SourceChEMBL;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O14965 AURKA Homo sapiens Human PF00069 7.8 IC50 ChEMBL
O75716 STK16 Homo sapiens Human PF00069 7.8 pIC50 TTD_MultiTarget
Q96GD4 AURKB Homo sapiens Human PF00069 6.3 IC50 ChEMBL