Molecule Details
InChIKeySWIHLLNXGOJYRM-WHOHXGKFSA-N
Compound Name(2S)-2-fluoro-2-[[(2S,5R)-3-methyl-7-oxo-2-[[(2S)-pyrrolidin-2-yl]methoxycarbamoyl]-1,6-diazabicyclo[3.2.1]oct-3-en-6-yl]oxy]acetic acid
Canonical SMILESCC1=C[C@@H]2CN(C(=O)N2O[C@@H](F)C(=O)O)[C@@H]1C(=O)NOC[C@@H]1CCCN1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.38
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P62593 bla Escherichia coli Pathogen PF13354 6.7 IC50 BindingDB
P00811 ampC Escherichia coli (strain K12) Pathogen PF00144 6.4 IC50 ChEMBL;BindingDB
Q6XEC0 OXA-48 Klebsiella pneumoniae Pathogen PF00905 6.1 IC50 BindingDB