Molecule Details
InChIKeySWHALWMKROAPPG-UHFFFAOYSA-N
Compound NameN-[4-[3-(cyclopropylmethyl)-7-fluoro-2-methylbenzimidazol-5-yl]-5-fluoropyrimidin-2-yl]-5,6,7,8-tetrahydro-1,6-naphthyridin-2-amine
Canonical SMILESCc1nc2c(F)cc(-c3nc(Nc4ccc5c(n4)CCNC5)ncc3F)cc2n1CC1CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.87
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P11802 CDK4 Homo sapiens Human PF00069 8.4 IC50 ChEMBL;BindingDB
Q00534 CDK6 Homo sapiens Human PF00069 8.2 IC50 ChEMBL;BindingDB
P24941 CDK2 Homo sapiens Human PF00069 7.0 IC50 ChEMBL;BindingDB