Molecule Details
InChIKeySWGQDPWKPYZEEH-SFHVURJKSA-N
Canonical SMILESCN(C)CCN[C@H](C(=O)NCc1cc(C(F)(F)F)cc(C(F)(F)F)c1)c1ccc(F)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL6.15
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P25103 TACR1 Homo sapiens Human PF00001 6.2 IC50 ChEMBL;BindingDB
P41597 CCR2 Homo sapiens Human PF00001 6.1 IC50 ChEMBL;BindingDB