Molecule Details
InChIKeySVYGTBODIFTCOZ-UHFFFAOYSA-N
Compound Namen-[6-(2-Fluorophenyl)-5-(3-fluoropyridin-4-yl)pyrazin-2-yl]cyclopropane-carboxamide
Canonical SMILESO=C(Nc1cnc(-c2ccncc2F)c(-c2ccccc2F)n1)C1CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.7
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P29275 ADORA2B Homo sapiens Human PF00001 9.2 Ki ChEMBL;BindingDB
P29274 ADORA2A Homo sapiens Human PF00001 7.0 Ki ChEMBL;BindingDB
P30542 ADORA1 Homo sapiens Human PF00001 6.9 Ki ChEMBL;BindingDB