Molecule Details
InChIKeySVOBVHOTNXSTLW-UHFFFAOYSA-N
Compound Name2-(N-Methyl-guanidino)-N-[4-(4-sulfamoyl-phenylamino)-pyrimidin-2-yl]-acetamide
Canonical SMILESCN(CC(=O)Nc1nccc(Nc2ccc(S(N)(=O)=O)cc2)n1)C(=N)N
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.64
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P00918 CA2 Homo sapiens Human PF00194 7.8 Ki ChEMBL;BindingDB
P18505 GABRB1 Homo sapiens Human PF02931 PF02932 7.8 pIC50 TTD_MultiTarget
P00915 CA1 Homo sapiens Human PF00194 7.3 Ki ChEMBL;BindingDB