Molecule Details
InChIKeySVLAHMNAIPTSSR-UHFFFAOYSA-N
Compound NameN-[4-(3-iodo-5-methylphenyl)-5-pyridin-4-yl-1,3-thiazol-2-yl]pyridine-3-carboxamide
Canonical SMILESCc1cc(I)cc(-c2nc(NC(=O)c3cccnc3)sc2-c2ccncc2)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.34
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P0DMS8 ADORA3 Homo sapiens Human PF00001 8.2 Ki ChEMBL;BindingDB
P35462 DRD3 Homo sapiens Human PF00001 6.5 Ki ChEMBL;BindingDB