Molecule Details
InChIKeySUXRXYKUAHNUAX-CLYVBNDRSA-N
Canonical SMILESCc1ccc(-c2cc(C(=O)N[C@H](C)c3ccc(F)cn3)cc(C3=NO[C@H](c4ccccn4)C3)c2)nc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL6.81
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P56373 P2RX3 Homo sapiens Human PF00864 7.6 IC50 ChEMBL;BindingDB
P22309 UGT1A1 Homo sapiens Human PF00201 6.0 IC50 ChEMBL;BindingDB