Molecule Details
InChIKeySURYSMJVQLKAOF-UHFFFAOYSA-N
Compound Name6-[3-(4-pyridin-2-yl-1,4-diazepan-1-yl)propoxy]-3,4-dihydro-1H-quinolin-2-one
Canonical SMILESO=C1CCc2cc(OCCCN3CCCN(c4ccccn4)CC3)ccc2N1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.34
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P31645 SLC6A4 Homo sapiens Human PF03491 PF00209 6.6 Ki ChEMBL;BindingDB
P08908 HTR1A Homo sapiens Human PF00001 6.4 Ki ChEMBL;BindingDB
P34969 HTR7 Homo sapiens Human PF00001 6.0 Ki ChEMBL;BindingDB