Molecule Details
InChIKeySUQBHZSJXAKKQX-MSQADJIASA-N
Compound NameN-[(2S)-1-[[(2S)-1-[[(3S)-1-(3-acetylanilino)-5-methyl-1,2-dioxohexan-3-yl]amino]-3-(4-methoxyphenyl)-1-oxopropan-2-yl]amino]-1-oxopropan-2-yl]-5-(4-acetylphenyl)furan-2-carboxamide
Canonical SMILESCOc1ccc(C[C@H](NC(=O)[C@H](C)NC(=O)c2ccc(-c3ccc(C(C)=O)cc3)o2)C(=O)N[C@@H](CC(C)C)C(=O)C(=O)Nc2cccc(C(C)=O)c2)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.95
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P28062 PSMB8 Homo sapiens Human PF00227 7.6 IC50 ChEMBL;BindingDB
P49721 PSMB2 Homo sapiens Human PF00227 6.9 IC50 ChEMBL;BindingDB
P20618 PSMB1 Homo sapiens Human PF00227 6.4 IC50 ChEMBL;BindingDB