Molecule Details
InChIKeySUODWKMMJQIJQB-XDJLXXALSA-N
Compound Name(1R)-2-[2-[(1S)-1-(4-chlorophenyl)ethyl]-3,3-dioxo-1,4-dihydroimidazo[5,1-d][1,2,5]thiadiazin-4-yl]-1-phenylethanol
Canonical SMILESC[C@@H](c1ccc(Cl)cc1)N1Cc2cncn2C(C[C@@H](O)c2ccccc2)S1(=O)=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.26
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P19099 CYP11B2 Homo sapiens Human PF00067 8.6 IC50 ChEMBL;BindingDB
P15538 CYP11B1 Homo sapiens Human PF00067 6.6 IC50 ChEMBL;BindingDB
P08684 CYP3A4 Homo sapiens Human PF00067 6.5 IC50 ChEMBL;BindingDB