Molecule Details
InChIKeySUIWTHQZBYYCGP-UHFFFAOYSA-N
Compound Name3-N-(1,3-dimethyl-2-oxoquinolin-6-yl)-1-N-hydroxy-4-methoxybenzene-1,3-dicarboxamide
Canonical SMILESCOc1ccc(C(=O)NO)cc1C(=O)Nc1ccc2c(c1)cc(C)c(=O)n2C
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.47
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9BY41 HDAC8 Homo sapiens Human PF00850 7.2 IC50 ChEMBL;BindingDB
Q9UBN7 HDAC6 Homo sapiens Human PF00850 PF02148 6.2 IC50 ChEMBL;BindingDB
P55201 BRPF1 Homo sapiens Human PF00439 PF10513 PF13831 PF00855 PF13832 6.1 Kd ChEMBL;BindingDB