Molecule Details
InChIKeySUHLJVHSQCIBRD-UHFFFAOYSA-N
Compound Name5-{5-[4-(3-Chloro-phenyl)-3-oxo-piperazin-1-ylmethyl]-imidazol-1-ylmethyl}-2-phenoxy-benzonitrile
Canonical SMILESN#Cc1cc(Cn2cncc2CN2CCN(c3cccc(Cl)c3)C(=O)C2)ccc1Oc1ccccc1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.4
SourceChEMBL;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P49354 FNTA Homo sapiens Human PF01239 8.1 pIC50 TTD_MultiTarget
P49356 FNTB Homo sapiens Human PF00432 8.1 IC50 ChEMBL
P53609 PGGT1B Homo sapiens Human PF00432 6.1 IC50 ChEMBL