Molecule Details
InChIKeySTWDLMHONRHMTF-UHFFFAOYSA-N
Compound Name5-(2,6-difluorophenyl)-3-[6-(4-methylidenepiperidin-3-yl)oxypyrazin-2-yl]-1H-indazole
Canonical SMILESC=C1CCNCC1Oc1cncc(-c2n[nH]c3ccc(-c4c(F)cccc4F)cc23)n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.31
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P11309 PIM1 Homo sapiens Human PF00069 8.5 IC50 ChEMBL;BindingDB
Q86V86 PIM3 Homo sapiens Human PF00069 8.4 IC50 ChEMBL;BindingDB
Q9P1W9 PIM2 Homo sapiens Human PF00069 8.0 IC50 ChEMBL;BindingDB