Molecule Details
InChIKeySTJJPAKEFZQZGB-UHFFFAOYSA-N
Compound Name7-Chloro-4-oxo-1-phenyl-3-[4-(piperazine-1-sulfonyl)-benzyl]-1,4-dihydroquinoline-2-carboxylic acid methyl ester
Canonical SMILESCOC(=O)c1c(Cc2ccc(S(=O)(=O)N3CCNCC3)cc2)c(=O)c2ccc(Cl)cc2n1-c1ccccc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.94
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P45983 MAPK8 Homo sapiens Human PF00069 7.5 IC50 ChEMBL;BindingDB
P45984 MAPK9 Homo sapiens Human PF00069 7.3 IC50 ChEMBL;BindingDB
P53779 MAPK10 Homo sapiens Human PF00069 6.0 IC50 ChEMBL