Molecule Details
InChIKeySTIKULJYVCUQJQ-UHFFFAOYSA-N
Compound Name6-Chloro-11-[2-[4-(2-methoxyphenyl)piperazin-1-yl]ethylamino]-4-methyl-4,5,9,10-tetrazatricyclo[7.4.0.02,7]trideca-1,5,7,10,12-pentaen-3-one
Canonical SMILESCOc1ccccc1N1CCN(CCNc2ccc3c4c(=O)n(C)nc(Cl)c4cn3n2)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.43
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P35348 ADRA1A Homo sapiens Human PF00001 9.0 Ki ChEMBL;BindingDB
P25100 ADRA1D Homo sapiens Human PF00001 8.5 Ki ChEMBL;BindingDB
P35368 ADRA1B Homo sapiens Human PF00001 7.8 Ki ChEMBL;BindingDB