Molecule Details
InChIKeySSXRGZQGLUZVSY-UHFFFAOYSA-N
Compound Name3-amino-N-(3-pyridyl)-6-(4-sulfamoylphenyl)pyrazine-2-carboxamide
Canonical SMILESNc1ncc(-c2ccc(S(N)(=O)=O)cc2)nc1C(=O)Nc1cccnc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)4
Pfam Stratification Cross-Family
Avg pChEMBL7.23
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (4)
Target Gene Organism Category Pfam pChEMBL Type Source
P49841 GSK3B Homo sapiens Human PF00069 7.9 Ki ChEMBL;BindingDB
O96020 CCNE2 Homo sapiens Human PF02984 PF00134 7.0 Ki ChEMBL
P24864 CCNE1 Homo sapiens Human PF02984 PF00134 7.0 Ki ChEMBL
P24941 CDK2 Homo sapiens Human PF00069 7.0 Ki ChEMBL