Molecule Details
InChIKeySSVPMKGPRCBPJY-UHFFFAOYSA-N
Compound Name3-Methyl-4-[5-[8-[(3-methyl-2-pyridinyl)methyl]-2,4-dioxo-1-pyrazin-2-yl-1,3,8-triazaspiro[4.5]decan-3-yl]-2-pyridinyl]benzoic acid
Canonical SMILESCc1cc(C(=O)O)ccc1-c1ccc(N2C(=O)N(c3cnccn3)C3(CCN(Cc4ncccc4C)CC3)C2=O)cn1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.46
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q96KS0 EGLN2 Homo sapiens Human PF13640 9.0 IC50 ChEMBL;BindingDB
Q9GZT9 EGLN1 Homo sapiens Human PF13640 PF01753 9.0 IC50 ChEMBL;BindingDB
Q9H6Z9 EGLN3 Homo sapiens Human PF13640 7.4 IC50 ChEMBL;BindingDB