Molecule Details
InChIKeySSBAFVYFCTXULM-UHFFFAOYSA-N
Compound Name8-(2-aminopyridin-4-yl)-7-(4-fluorophenyl)-2-((3-fIuoropyridin-2-yl)methyl)-[1,2,4]triazolo[1,5-c]pyrmidin-5-amine
Canonical SMILESNc1cc(-c2c(-c3ccc(F)cc3)nc(N)n3nc(Cc4ncccc4F)nc23)ccn1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.63
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P30542 ADORA1 Homo sapiens Human PF00001 8.1 IC50 ChEMBL;BindingDB
P29275 ADORA2B Homo sapiens Human PF00001 7.4 IC50 ChEMBL;BindingDB
P29274 ADORA2A Homo sapiens Human PF00001 7.4 IC50 ChEMBL;BindingDB