Molecule Details
InChIKeySQMSKBYHTUAWDC-UHFFFAOYSA-N
Compound Name2-[[3-(2-aminoethyl)-1H-indol-5-yl]oxy]-1-[4-[1-[2-[[3-(2-aminoethyl)-1H-indol-5-yl]oxy]acetyl]piperidin-4-yl]piperidin-1-yl]ethanone
Canonical SMILESNCCc1c[nH]c2ccc(OCC(=O)N3CCC(C4CCN(C(=O)COc5ccc6[nH]cc(CCN)c6c5)CC4)CC3)cc12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL9.21
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P28222 HTR1B Homo sapiens Human PF00001 9.7 Ki ChEMBL;BindingDB
P28221 HTR1D Homo sapiens Human PF00001 9.6 Ki ChEMBL;BindingDB
P08908 HTR1A Homo sapiens Human PF00001 8.4 Ki ChEMBL;BindingDB