Molecule Details
InChIKeySPRLNKQKOJIGIN-UHFFFAOYSA-N
Compound Name1-(5-Fluoro-2-methoxyphenyl)-4-[4-(2-methoxyphenyl)piperazin-1-yl]pyrazolo[5,4-d]pyrimidine
Canonical SMILESCOc1ccccc1N1CCN(c2ncnc3c2cnn3-c2cc(F)ccc2OC)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.69
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P11166 SLC2A1 Homo sapiens Human PF00083 7.5 IC50 ChEMBL;BindingDB
P11169 SLC2A3 Homo sapiens Human PF00083 6.5 IC50 ChEMBL;BindingDB
P11168 SLC2A2 Homo sapiens Human PF00083 6.1 IC50 ChEMBL;BindingDB