Molecule Details
InChIKeySPEKKKWCEBGMGP-UHFFFAOYSA-N
Compound NameN-(2-bromoprop-2-en-1-yl)-N-{6-cyano-1-[(1-methyl-1H-imidazol-5-yl)methyl]-1,2,3,4-tetrahydroquinolin-3-yl}-1-methyl-1H-imidazole-4-sulfonamide
Canonical SMILESC=C(Br)CN(C1Cc2cc(C#N)ccc2N(Cc2cncn2C)C1)S(=O)(=O)c1cn(C)cn1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL9.4
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q5E175 rhlE Aliivibrio fischeri (strain ATCC 700601 / ES114) Pathogen PF00270 PF00271 9.4 IC50 BindingDB
Q5EI73 Plasmodium falciparum Pathogen PF01239 9.4 IC50 ChEMBL