Molecule Details
InChIKeySOHWYEVCBPDAIO-UHFFFAOYSA-N
Compound Name4-methoxy-2-methyl-5-(2-methyl-4-pyridinyl)-7H-pyrrolo[2,3-d]pyrimidine
Canonical SMILESCOc1nc(C)nc2[nH]cc(-c3ccnc(C)c3)c12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.15
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q13627 DYRK1A Homo sapiens Human PF00069 7.5 IC50 ChEMBL;BindingDB
Q9Y463 DYRK1B Homo sapiens Human PF00069 7.4 IC50 ChEMBL;BindingDB
Q92630 DYRK2 Homo sapiens Human PF00069 6.5 IC50 ChEMBL;BindingDB