Molecule Details
InChIKeySMWIKHQGVFQHQV-UHFFFAOYSA-N
Canonical SMILESNS(=O)(=O)NCc1nnc(C(c2nc3ccc(-c4ccc(C(=O)N5CCOCC5)c(Cl)c4)cc3s2)S(=O)(=O)Cc2ccccc2)o1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.08
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9Y5X9 LIPG Homo sapiens Human PF00151 PF01477 7.2 IC50 ChEMBL;BindingDB
P11150 LIPC Homo sapiens Human PF00151 PF01477 6.9 IC50 ChEMBL;BindingDB