Molecule Details
InChIKeySMRAUEYCFQUGMY-UHFFFAOYSA-N
Compound Name4-[8-(Dimethylamino)-3-oxo-2-phenyl-[1,2,4]triazolo[4,3-a]pyrazin-6-yl]benzenesulfonamide
Canonical SMILESCN(C)c1nc(-c2ccc(S(N)(=O)=O)cc2)cn2c(=O)n(-c3ccccc3)nc12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.38
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O43570 CA12 Homo sapiens Human PF00194 6.5 Ki ChEMBL;BindingDB
P30542 ADORA1 Homo sapiens Human PF00001 6.4 Ki ChEMBL;BindingDB
P00918 CA2 Homo sapiens Human PF00194 6.3 Ki ChEMBL;BindingDB