Molecule Details
InChIKeySMLFVHZWGKWRSD-UHFFFAOYSA-N
Compound Name4-bromo-2-methyl-7,8,9,10-tetrahydro-6H-cyclohepta[b]quinoline-11-carboxylic acid
Canonical SMILESCc1cc(Br)c2nc3c(c(C(=O)O)c2c1)CCCCC3
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.43
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P04156 PRNP Homo sapiens Human PF00377 PF11587 PF03991 6.8 IC50 ChEMBL;BindingDB
P37231 PPARG Homo sapiens Human PF00104 PF12577 PF00105 6.2 IC50 ChEMBL
Q9Y618 NCOR2 Homo sapiens Human PF15784 PF00249 6.2 IC50 ChEMBL;BindingDB