Molecule Details
InChIKeySLRQWILFIQMPFZ-UHFFFAOYSA-N
Compound Name8-bromo-2-[1-(4-methylpiperazin-1-yl)ethyl]-3H-[1]benzofuro[3,2-d]pyrimidin-4-one
Canonical SMILESCC(c1nc2c(oc3ccc(Br)cc32)c(=O)[nH]1)N1CCN(C)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.19
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P11309 PIM1 Homo sapiens Human PF00069 7.8 IC50 ChEMBL;BindingDB
Q86V86 PIM3 Homo sapiens Human PF00069 7.5 IC50 ChEMBL;BindingDB
Q9P1W9 PIM2 Homo sapiens Human PF00069 6.3 IC50 ChEMBL;BindingDB