Target not found.
Molecule Details
InChIKeySLORTXJSOVPUPP-UHFFFAOYSA-N
Compound NameN-[5-fluoro-4-(8-fluoro-4-propan-2-yl-2,3-dihydro-1,4-benzoxazin-6-yl)pyrimidin-2-yl]-5-methyl-6,7-dihydro-4H-pyrazolo[1,5-a]pyrazin-2-amine
Canonical SMILESCC(C)N1CCOc2c(F)cc(-c3nc(Nc4cc5n(n4)CCN(C)C5)ncc3F)cc21
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL8.15
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P11802 CDK4 Homo sapiens Human PF00069 8.8 IC50 ChEMBL;BindingDB
Q00534 CDK6 Homo sapiens Human PF00069 8.5 IC50 ChEMBL;BindingDB
P07333 CSF1R Homo sapiens Human PF00047 PF25305 PF07714 7.2 IC50 ChEMBL;BindingDB