Molecule Details
InChIKeySLOIJUIDHUKLRX-UHFFFAOYSA-N
Compound Name3-(6-Amino-5-(1-oxo-1,2,3,4-tetrahydroisoquinolin-6-yl)pyridin-3-yl)benzonitrile
Canonical SMILESN#Cc1cccc(-c2cnc(N)c(-c3ccc4c(c3)CCNC4=O)c2)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.7
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q13043 STK4 Homo sapiens Human PF11629 PF00069 6.9 IC50 ChEMBL;BindingDB
Q13188 STK3 Homo sapiens Human PF11629 PF00069 6.9 IC50 ChEMBL;BindingDB
Q9Y6E0 STK24 Homo sapiens Human PF20929 PF00069 6.3 IC50 ChEMBL;BindingDB