Molecule Details
InChIKeySJTLDCMGGRCPJQ-UHFFFAOYSA-N
Compound Name3-[[4-(2-amino-1,3-benzothiazol-4-yl)-2-sulfamoyl-3-(2H-tetrazol-5-yl)phenyl]sulfonylamino]propyl-trimethylazanium
Canonical SMILESC[N+](C)(C)CCCNS(=O)(=O)c1ccc(-c2cccc3sc(N)nc23)c(-c2nnn[nH]2)c1S(N)(=O)=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL10.05
SourceBindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
C7C422 blaNDM-1 Klebsiella pneumoniae Pathogen PF00753 10.5 IC50 BindingDB
Q2QC95 blaoxa-10 Klebsiella pneumoniae Pathogen PF00905 10.0 IC50 BindingDB
P52699 Serratia marcescens Pathogen PF00753 9.7 IC50 BindingDB