Molecule Details
InChIKeySJIMFBGRZWUIGY-BGXLBEBNSA-N
Compound Namecyclo[N(Me)Ala-Tyr-D-N(Me)Trp-N(Me)Lys-Val-N(Me)Phe]
Canonical SMILESCC(C)[C@@H]1NC(=O)[C@H](CCCCN)N(C)C(=O)[C@@H](Cc2c[nH]c3ccccc23)N(C)C(=O)[C@H](Cc2ccc(O)cc2)NC(=O)[C@H](C)N(C)C(=O)[C@H](Cc2ccccc2)N(C)C1=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.88
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P30874 SSTR2 Homo sapiens Human PF00001 7.4 IC50 ChEMBL;BindingDB
P32745 SSTR3 Homo sapiens Human PF00001 6.7 IC50 ChEMBL;BindingDB
P35346 SSTR5 Homo sapiens Human PF00001 6.6 IC50 ChEMBL;BindingDB