Molecule Details
InChIKeySIUKGJQBSLZIDB-UNOMPAQXSA-N
Compound Name(5Z)-5-[(4-phenylmethoxyphenyl)methylidene]-3-[2-[3-(trifluoromethyl)-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl]acetyl]-1,3-thiazolidine-2,4-dione
Canonical SMILESO=C(CN1CCn2c(nnc2C(F)(F)F)C1)N1C(=O)S/C(=C\c2ccc(OCc3ccccc3)cc2)C1=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.73
SourceChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P27487 DPP4 Homo sapiens Human PF00930 PF00326 6.9 IC50 ChEMBL
P18031 PTPN1 Homo sapiens Human PF00102 6.8 IC50 ChEMBL
P0DUB6 AMY1A Homo sapiens Human PF00128 PF02806 6.5 IC50 ChEMBL