Molecule Details
InChIKeySIPQEKQXLUBVAY-GJZGRUSLSA-N
Compound Name1-Aminomethyl-6-bromo-3-phenyl-isochroman-5-ol; hydrochloride
Canonical SMILESNC[C@@H]1O[C@H](c2ccccc2)Cc2c1ccc(Br)c2O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)4
Pfam Stratification Homologous
Avg pChEMBL6.51
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (4)
Target Gene Organism Category Pfam pChEMBL Type Source
P28335 HTR2C Homo sapiens Human PF00001 6.7 Ki ChEMBL;BindingDB
P08913 ADRA2A Homo sapiens Human PF00001 6.4 Ki ChEMBL;BindingDB
P18089 ADRA2B Homo sapiens Human PF00001 6.4 Ki ChEMBL
P18825 ADRA2C Homo sapiens Human PF00001 6.4 Ki ChEMBL