Molecule Details
InChIKeySHVVVMSMELBKDU-VKVKMMGJSA-N
Compound Name4-[4-[(Z)-[[4-(6-chloro-2-oxochromen-3-yl)-1,3-thiazol-2-yl]hydrazinylidene]methyl]-3-(4-chlorophenyl)pyrazol-1-yl]benzenesulfonamide
Canonical SMILESNS(=O)(=O)c1ccc(-n2cc(/C=N\Nc3nc(-c4cc5cc(Cl)ccc5oc4=O)cs3)c(-c3ccc(Cl)cc3)n2)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.69
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O43570 CA12 Homo sapiens Human PF00194 8.5 Ki ChEMBL;BindingDB
Q16790 CA9 Homo sapiens Human PF00194 7.5 Ki ChEMBL;BindingDB
P00918 CA2 Homo sapiens Human PF00194 7.0 Ki ChEMBL;BindingDB