Molecule Details
InChIKeySHKOYYABTMCHBH-BGYRXZFFSA-N
Compound Name1-[[2-(2-chloro-6-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl]-N-[3-[(3S,5R)-3,5-dimethylpiperidin-1-yl]propyl]piperidine-4-carboxamide
Canonical SMILESCc1cccc(Cl)c1-c1nc(CN2CCC(C(=O)NCCCN3C[C@H](C)C[C@H](C)C3)CC2)c(C)o1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.32
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P41595 HTR2B Homo sapiens Human PF00001 6.4 Ki ChEMBL;BindingDB
P25021 HRH2 Homo sapiens Human PF00001 6.3 Ki ChEMBL;BindingDB
P18825 ADRA2C Homo sapiens Human PF00001 6.2 Ki ChEMBL;BindingDB