Molecule Details
InChIKeySGVBVAOVXTWIJT-UHFFFAOYSA-N
Compound Name1-(4-((2-((3-(2,5,8,11,14-Pentaoxahexadecan-16-yloxy)-5-methoxyphenyl)amino)-pyrimidin-4-yl)oxy)naphthalen-1-yl)-3-(3-isopropyl-1-(p-tolyl)-1H-pyrazol-5-yl)urea
Canonical SMILESCOCCOCCOCCOCCOCCOc1cc(Nc2nccc(Oc3ccc(NC(=O)Nc4cc(C(C)C)nn4-c4ccc(C)cc4)c4ccccc34)n2)cc(OC)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.94
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P12931 SRC Homo sapiens Human PF07714 PF00017 PF00018 8.4 IC50 ChEMBL;BindingDB
P43405 SYK Homo sapiens Human PF07714 PF00017 7.9 IC50 ChEMBL;BindingDB
P53778 MAPK12 Homo sapiens Human PF00069 7.5 IC50 ChEMBL;BindingDB