Molecule Details
InChIKeySGRYPBLWIZFTHU-UHFFFAOYSA-N
Compound Name3-((3,3-dimethylmorpholino)methyl)-N-(6-methyl-3-(1H-pyrazol-4-yl)imidazo[1,2-a]pyrazin-8-yl)isothiazol-5-amine
Canonical SMILESCc1cn2c(-c3cn[nH]c3)cnc2c(Nc2cc(CN3CCOCC3(C)C)ns2)n1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL7.41
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
O75716 STK16 Homo sapiens Human PF00069 8.4 pIC50 TTD_MultiTarget
P06239 LCK Homo sapiens Human PF07714 PF00017 PF00018 6.4 IC50 ChEMBL;BindingDB