Molecule Details
InChIKeySFPAQPMKUYAZGZ-UHFFFAOYSA-N
Compound Name3-(1-(4-(4-Chloronaphthalen-1-ylamino)-4-oxobutyl)-1H-1,2,3-triazol-4-yl)-6-hydroxy-2-para-tolylbenzofuran-5-carboxylic Acid
Canonical SMILESCc1ccc(-c2oc3cc(O)c(C(=O)O)cc3c2-c2cn(CCCC(=O)Nc3ccc(Cl)c4ccccc34)nn2)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.51
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P18031 PTPN1 Homo sapiens Human PF00102 6.7 IC50 ChEMBL;BindingDB
P29350 PTPN6 Homo sapiens Human PF00017 PF00102 6.4 IC50 ChEMBL;BindingDB
Q9Y2R2 PTPN22 Homo sapiens Human PF00102 6.4 IC50 ChEMBL;BindingDB